SB-277011 hydrochloride
更新时间:2020-12-18 22:54:27
采购访问:1次
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常用名 |
SB-277011 hydrochloride |
CAS号 |
215804-67-4 |
价格 |
$需询单/250mg $需询单/100mg $需询单/1g |
纯度 |
98.0% |
备货期 |
3天 |
库存 |
现货 |
产品网页 |
http://www.dcchemicals.com/product_show-SB-277011_hydrochloride.html |
产品详情(用途,包装等) SB-277011 hydrochloride (SB-277011A hydrochloride) is a potent, selective, orally bioavailable and brain penetrate?dopamine D3?receptor (D3R)?antagonist with Ki values of 10.7?nM and?11.2 nM?at?rodent and human?D3R, respectively. SB-277011 hydrochloride displays 80- to 100-fold selectivity over other dopamine receptors with?pKis of 8.0, 6.0, <5.2, and 5.9 for D3, D2, 5-HT1B, and 5-HT1D receptors, respectively. |
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