SCH 23390 maleate
更新时间:2020-12-18 22:54:27
采购访问:1次
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常用名 |
SCH 23390盐酸盐 |
CAS号 |
87134-87-0 |
价格 |
$500.0/100mg $1000.0/250mg $2000.0/1g |
纯度 |
98.0% |
备货期 |
3天 |
库存 |
现货 |
产品网页 |
http://www.dcchemicals.com/product_show-SCH_23390_maleate.html |
产品详情(用途,包装等) SCH-23390 is a potent dopamine receptor antagonist (Ki values are 0.2 nM and 0.3 nM at D1 and D5 receptor sub-types, respectively). SCH-23390 is also an agonist at 5-HT1C and 5-HT2C receptors in vitro (Ki values are 6.3 nM and 9.3 nM respectively). It blocks quinpirole-induced Kir3 (GIRK) currents (EC50 = 268 nM) independently of receptors. |
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